Org-12962
CAS No. 132834-56-1
Org-12962 ( —— )
产品货号. M26777 CAS No. 132834-56-1
Org-12962 is an effective and selective 5-HT2C receptor agonist pEC50: 7.01). Org-12962 shows antiaversive effects in a rat model of panic-like anxiety.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥332 | 有现货 |
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10MG | ¥535 | 有现货 |
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25MG | ¥794 | 有现货 |
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50MG | ¥1118 | 有现货 |
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100MG | ¥1596 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Org-12962
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Org-12962 is an effective and selective 5-HT2C receptor agonist pEC50: 7.01). Org-12962 shows antiaversive effects in a rat model of panic-like anxiety.
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产品描述Org-12962 is an effective and selective 5-HT2C receptor agonist pEC50: 7.01). Org-12962 shows antiaversive effects in a rat model of panic-like anxiety. Org-12962 also shows high effacy for the 5-HT2A and 5-HT2B receptors (pEC50s: 6.38 and 6.28, respectively).(In Vivo):Org-12962 is dissolved or microsuspended in 0.3% v/v Tween 80 in physiological saline (NaCl 0.9%). Org-12962 (intraperitoneal injection; 0.3-3.2 mg/kg) obviously enhances the postinjection frequency thresholds for self-interruption (F3.71=11.40) .
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同义词——
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体HCV; Nucleoside Antimetabolite/Analog
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研究领域——
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适应症——
化学信息
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CAS Number132834-56-1
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分子量265.7
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分子式C10H11ClF3N3
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纯度>98% (HPLC)
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溶解度——
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SMILESFC(F)(F)c1ccc(nc1Cl)N1CCNCC1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Steven S Carroll, et al. Inhibition of hepatitis C virus RNA replication by 2'-modified nucleoside analogs. J Biol Chem. 2003 Apr 4;278(14):11979-84
产品手册
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