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Ogerin
CAS No. 1309198-71-7
Ogerin ( —— )
产品货号. M23467 CAS No. 1309198-71-7
Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥356 | 有现货 |
|
| 5MG | ￥551 | 有现货 |
|
| 10MG | ￥948 | 有现货 |
|
| 25MG | ￥1936 | 有现货 |
|
| 50MG | ￥3248 | 有现货 |
|
| 100MG | ￥4836 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Ogerin
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice.
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产品描述Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and antagonist activity (Ki, 220 nM) at A2A receptor and weak antagonist activity (Ki, 736 nM) at 5-HT2B receptor.
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同义词——
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT2B;A2A;GPR68
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研究领域——
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适应症——
化学信息
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CAS Number1309198-71-7
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分子量307.4
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分子式C17H17N5O
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纯度>98% (HPLC)
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溶解度DMSO:250 mg/mL (813.40 mM; Need ultrasonic)
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SMILESOCC1=C(C2=NC(N)=NC(NCC3=CC=CC=C3)=N2)C=CC=C1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Huang XP, et al. Allosteric ligands for the pharmacologically dark receptors GPR68 and GPR65. Nature. 2015 Nov 26;527(7579):477-83.
产品手册
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