NIH-12848
CAS No. 959551-10-1
NIH-12848 ( NIH-12848;NCGC00012848-02. )
产品货号. M17694 CAS No. 959551-10-1
NIH-12848 is a putative inhibitor of phosphatidylinositol 5-phosphate 4-kinase γ (PI5P4Kγ) with an IC50 of 1 μM.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥437 | 有现货 |
|
5MG | ¥689 | 有现货 |
|
10MG | ¥988 | 有现货 |
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25MG | ¥1928 | 有现货 |
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50MG | ¥3394 | 有现货 |
|
100MG | ¥4836 | 有现货 |
|
500MG | ¥10368 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称NIH-12848
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述NIH-12848 is a putative inhibitor of phosphatidylinositol 5-phosphate 4-kinase γ (PI5P4Kγ) with an IC50 of 1 μM.
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产品描述NIH-12848 is a putative phosphatidylinositol 5-phosphate 4-kinase γ (PI5P4Kγ) inhibitor. NIH-12848 inhibited PI5P4Kγ with an IC50 of approximately 1 μM but did not inhibit the α and β PI5P4K isoforms at concentrations up to 100 μM. NIH-12848 is a potentially powerful tool for exploring the cell physiology of PI5P4Ks.
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同义词NIH-12848;NCGC00012848-02.
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通路GPCR/G Protein
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靶点Neurokinin Receptor
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受体PI5P4Kγ
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研究领域——
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适应症——
化学信息
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CAS Number959551-10-1
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分子量385.41
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分子式C20H14F3N3S
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纯度98%
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溶解度DMSO : ≥ 28 mg/mL; 72.65 mM
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SMILESFC(F)(F)c1ccccc1c1nc2ccccc2c(NCc2cccs2)n1
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化学全称N-(thiophen-2-ylmethyl)-2-(2-(trifluoromethyl)phenyl)quinazolin-4-amine
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Clarke JH,et al.Biochem J. 2015 Mar 1;466(2):359-67.
产品手册
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