N-Acetyl-Calicheamicin
CAS No. 108212-76-6
N-Acetyl-Calicheamicin ( N-Acetyl-Calicheamicin γ;N-Acetyl-γ-calicheamicin )
产品货号. M10325 CAS No. 108212-76-6
N-Acetyl-Calicheamicin is a enediyne antitumor antibiotic; targets DNA and causes strand scission.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥9153 | 有现货 |
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10MG | ¥12312 | 有现货 |
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25MG | ¥18225 | 有现货 |
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50MG | ¥24057 | 有现货 |
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100MG | 获取报价 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称N-Acetyl-Calicheamicin
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述N-Acetyl-Calicheamicin is a enediyne antitumor antibiotic; targets DNA and causes strand scission.
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产品描述N-Acetyl-Calicheamicin is a enediyne antitumor antibiotic; targets DNA and causes strand scission; a ADC payload in antibody drug conjugates development.
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同义词N-Acetyl-Calicheamicin γ;N-Acetyl-γ-calicheamicin
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通路GPCR/G Protein
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靶点Antibacterial
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受体Antibacterial
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研究领域Cancer
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适应症——
化学信息
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CAS Number108212-76-6
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分子量1410.39
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分子式C57H76IN3O22S4
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纯度>98% (HPLC)
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溶解度10 mM in DMSO
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SMILESCCN(C1COC(CC1OC)OC2C(C(C(OC2OC3C#CC=CC#CC4(CC(=O)C(=C3C4=CCSSSC)NC(=O)OC)O)C)NOC5CC(C(C(O5)C)SC(=O)C6=C(C(=C(C(=C6OC)OC)OC7C(C(C(C(O7)C)O)OC)O)I)C)O)O)C(=O)C
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化学全称Carbamic acid, [(1R,4Z,8S,13E)-8-[[2-O-[4-(acetylethylamino)-2,4-dideoxy-3-O-methyl-α-L-threo-pentopyranosyl]-4,6-dideoxy-4-[[[2,6-dideoxy-4-S-[4-[(6-deoxy-3-O-methyl-α-L-mannopyranosyl)oxy]-3-iodo-5,6-dimethoxy-2-methylbenzoyl]-4-thio-β-D-ribo-hexopyrano
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Stasi R, et al. Cancer Treat Rev. 2008 Feb;34(1):49-60.
2. Naito K, et al. Leukemia. 2000 Aug;14(8):1436-43.
3. Hills RK, et al. Lancet Oncol. 2014 Aug;15(9):986-96.
2. Naito K, et al. Leukemia. 2000 Aug;14(8):1436-43.
3. Hills RK, et al. Lancet Oncol. 2014 Aug;15(9):986-96.
产品手册
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