Mirodenafil
CAS No. 862189-95-5
Mirodenafil ( SK3530 )
产品货号. M22579 CAS No. 862189-95-5
Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.The pharmacoki-netics of mirodenafil were not significantly altered by this concurrent administration. Mirodenafil (50 or 100 mg), obviously improved erectile function and was well tolerated in a representative population of Korean men with broad-spectrum ED of various etiologies and severities.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥2446 | 有现货 |
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10MG | ¥3669 | 有现货 |
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25MG | ¥6051 | 有现货 |
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50MG | ¥8505 | 有现货 |
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100MG | ¥11502 | 有现货 |
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500MG | ¥22923 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Mirodenafil
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.The pharmacoki-netics of mirodenafil were not significantly altered by this concurrent administration. Mirodenafil (50 or 100 mg), obviously improved erectile function and was well tolerated in a representative population of Korean men with broad-spectrum ED of various etiologies and severities.
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产品描述Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.The pharmacoki-netics of mirodenafil were not significantly altered by this concurrent administration. Mirodenafil (50 or 100 mg), obviously improved erectile function and was well tolerated in a representative population of Korean men with broad-spectrum ED of various etiologies and severities. Mirodenafil administered with alcohol had a tolerability profile comparable to that of mirodenafil alone. The concurrent administration of mirodenafil with alcohol was not associated with clinically significant hemodynamic changes in these healthy male volunteers in Korea. The coadministration of ketoconazole and rifampicin resulted in significant changes in systemic exposure to mirodenafil, in these healthy Korean male volunteers.
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同义词SK3530
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通路Angiogenesis
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靶点PDE
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受体PDE5
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研究领域——
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适应症——
化学信息
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CAS Number862189-95-5
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分子量531.67
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分子式C26H37N5O5S
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纯度>98% (HPLC)
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溶解度——
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SMILESCCCOc1ccc(cc1-c1nc2c(CCC)cn(CC)c2c(=O)[nH]1)S(=O)(=O)N1CCN(CCO)CC1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Paick, J.S., et al., Efficacy and safety of mirodenafil, a new oral phosphodiesterase type 5 inhibitor, for treatment of erectile dysfunction. J Sex Med, 2008. 5(11): p. 2672-80.
产品手册
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