MKC-1
CAS No. 125313-92-0
MKC-1 ( —— )
产品货号. M28925 CAS No. 125313-92-0
MKC-1 is an orally bioavailable, small-molecule, bisindolylmaleimide cell cycle inhibitor with potential antineoplastic activity. MKC-1 and its metabolites inhibit tubulin polymerization, blocking the formation of the mitotic spindle.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥1725 | 有现货 |
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10MG | ¥2535 | 有现货 |
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25MG | ¥4390 | 有现货 |
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50MG | ¥6334 | 有现货 |
|
100MG | ¥8829 | 有现货 |
|
500MG | ¥17739 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称MKC-1
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述MKC-1 is an orally bioavailable, small-molecule, bisindolylmaleimide cell cycle inhibitor with potential antineoplastic activity. MKC-1 and its metabolites inhibit tubulin polymerization, blocking the formation of the mitotic spindle.
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产品描述MKC-1 is an orally bioavailable, small-molecule, bisindolylmaleimide cell cycle inhibitor with potential antineoplastic activity. MKC-1 and its metabolites inhibit tubulin polymerization, blocking the formation of the mitotic spindle.
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同义词——
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通路Apoptosis
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靶点Apoptosis
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受体——
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研究领域——
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适应症——
化学信息
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CAS Number125313-92-0
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分子量400.4
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分子式C22H16N4O4
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纯度>98% (HPLC)
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溶解度——
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SMILESCn1cc(C2=C(C(=O)NC2=O)c2cn(C)c3cc(ccc23)[N+]([O-])=O)c2ccccc12
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Hyland EE, et al. Unified Access to Pyrimidines and Quinazolines Enabled by N-N Cleaving Carbon Atom Insertion. J Am Chem Soc. 2022 Oct 26;144(42):19258-19264.
产品手册
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