MK-212 ( MK 212;MK212 )

产品货号. M15329 CAS No. 61655-58-1

A potent, selective 5-HT2C receptor agonist with IC50 of 20 nM in HEK293 cells-exppressed 5-HT2C, shows weakly activity for 5-HT2A.

纯度: >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

规格	价格/人民币	库存	数量
5MG	￥518	有现货
10MG	￥721	有现货
25MG	￥1725	有现货
50MG	￥3208	有现货
100MG	￥4771	有现货
500MG	￥10368	有现货
1G	获取报价	有现货

拼团产品询价大包装询价加入购物车

生物学信息

产品名称

MK-212
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

A potent, selective 5-HT2C receptor agonist with IC50 of 20 nM in HEK293 cells-exppressed 5-HT2C, shows weakly activity for 5-HT2A.
产品描述

A potent, selective 5-HT2C receptor agonist with IC50 of 20 nM in HEK293 cells-exppressed 5-HT2C, shows weakly activity for 5-HT2A; stimulates phosphoinositide hydrolysis in cerebral cortex, antagonizes the analgesia induced by either morphine or THIP in vivo.
同义词

MK 212;MK212
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT Receptor
研究领域

——
适应症

——

化学信息

CAS Number

61655-58-1
分子量

235.12
分子式

C8H11ClN4.HCl
纯度

>98% (HPLC)
溶解度

——
SMILES

ClC1=CN=CC(N2CCNCC2)=N1.[H]Cl
化学全称

6-Chloro-2-(1-piperazinyl)pyrazine hydrochloride

运输与储存

储存条件

(-20℃)
运输条件

With Ice Pack
稳定性

≥ 2 years

参考文献

1. Conn PJ, et al. J Pharmacol Exp Ther. 1987 Aug;242(2):552-7.
2. Hemrick-Luecke SK, et al. Eur J Pharmacol. 1996 Sep 12;311(2-3):207-11.
3. Jensen AA, et al. J Med Chem. 2013 Feb 14;56(3):1211-27.
4. Murray TF, et al. Eur J Pharmacol. 1983 Jun 3;90(2-3):179-84.

计算器

浓度计算器

摩尔计算器

分子量计算器

产品手册

关联产品

Elemicin

Elemicin is a constituent of several plant species' essential oils. It has anticholinergic effects in humans
Trimipramine maleate

Tricyclic antidepressant similar to IMIPRAMINE, but with more antihistaminic and sedative properties.
Dehydroaripiprazole

Dehydroaripiprazole is the active metabolite of aripiprazole. Aripiprazole is an antipsychotic drug, which is metabolized by CYP3A4 and CYP2D6 and mainly forms dehydroaripiprazole.

Product			Quantity Required*
Name *			E-mail Address *
Organization *			Phone Number
Remarks