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Galnon TFA

CAS No. 1217448-19-5

Galnon TFA ( —— )

产品货号. M37581 CAS No. 1217448-19-5

Galnon TFA 是一种选择性的非肽类的甘丙肽 GAL1 和 GAL2 受体激动剂,其 Ki 值分别为 11.7 和 34.1 μM。Galnon TFA 具有抗惊厥和抗焦虑作用。

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥1159 有现货
10MG ¥1720 有现货
25MG ¥2688 有现货
50MG ¥3636 有现货
100MG ¥4725 有现货
200MG ¥6210 有现货
500MG 获取报价 有现货
1G 获取报价 有现货
1 mL x 10 mM in DMSO ¥698 有现货

生物学信息

  • 产品名称
    Galnon TFA
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Galnon TFA 是一种选择性的非肽类的甘丙肽 GAL1 和 GAL2 受体激动剂,其 Ki 值分别为 11.7 和 34.1 μM。Galnon TFA 具有抗惊厥和抗焦虑作用。
  • 产品描述
    Galnon TFA is a selective and non-peptide agonist of galanin GAL1 and GAL2 receptor, with Kis of 11.7 and 34.1 μM respectively. Galnon TFA exhibits anticonvulsant and anxiolytic effects.
  • 体外实验
    ——
  • 体内实验
    ——
  • 同义词
    ——
  • 通路
    GPCR/G Protein
  • 靶点
    Neuropeptide Y Receptor
  • 受体
    Neuropeptide Y Receptor
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1217448-19-5
  • 分子量
    792.84
  • 分子式
    C42H47F3N4O8
  • 纯度
    >98% (HPLC)
  • 溶解度
    In Vitro:?DMSO 中的溶解度 : 125 mg/mL (157.66 mM; 超声助溶 )
  • SMILES
    C(C(O)=O)(F)(F)F.C(OC(N[C@@H](CC1CCCCC1)C(N[C@H](C(NC=2C=C3C(=CC2)C(C)=CC(=O)O3)=O)CCCCN)=O)=O)C4C=5C(C=6C4=CC=CC6)=CC=CC5
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Bartfai T, et, al. Galmic, a nonpeptide galanin receptor agonist, affects behaviors in seizure, pain, and forced-swim tests. Proc Natl Acad Sci U S A. 2004 Jul 13;101(28):10470-5.?
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