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NaV1.2/1.6 channel blocker-1
CAS No. 1199944-04-1
NaV1.2/1.6 channel blocker-1 ( —— )
产品货号. M36447 CAS No. 1199944-04-1
NaV1.2/1.6 channel blocker-1 是一种有效的 NaV1.2/1.6 channel 阻滞剂，抑制 rNaV1.6 和 hNaV1.2 的 IC50 值分别为 9.8 和 24.4 μM。NaV1.2/1.6 channel blocker-1 可用于全身性癫痫的研究。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥585 | 有现货 |
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| 10MG | ￥886 | 有现货 |
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| 25MG | ￥1739 | 有现货 |
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| 50MG | ￥2576 | 有现货 |
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| 100MG | ￥3717 | 有现货 |
|
| 200MG | ￥5292 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称NaV1.2/1.6 channel blocker-1
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述NaV1.2/1.6 channel blocker-1 是一种有效的 NaV1.2/1.6 channel 阻滞剂，抑制 rNaV1.6 和 hNaV1.2 的 IC50 值分别为 9.8 和 24.4 μM。NaV1.2/1.6 channel blocker-1 可用于全身性癫痫的研究。
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产品描述NaV1.2/1.6 channel blocker-1 is a potent NaV1.2/1.6 channel blocker, with IC50s of 9.8 and 24.4 μM for rNaV1.6 and hNaV1.2, respectively. NaV1.2/1.6 channel blocker-1 can be used for the research of generalized epilepsy.
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体外实验——
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体内实验——
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同义词——
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通路Membrane Transporter/Ion Channel
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靶点Sodium Channel
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受体Sodium Channel
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研究领域——
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适应症——
化学信息
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CAS Number1199944-04-1
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分子量258.34
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分子式C14H14N2OS
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纯度>98% (HPLC)
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溶解度——
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SMILESS=C1OC=2C=CC=CC2C3=NC(=C(N13)CCC)C
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
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A-317567
A-317567 (A317567) 是一种新型强效酸传感离子通道 (ASIC) 阻断剂，IC50 为 2-30 uM。
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Silperisone HCl
Silperisone HCl (RGH-5002) blocks sodium and calcium channels in cells, decreases excitability and contractility of muscle cells, reduces peripheral tone, and acts as a muscle relaxant and peripheral vasodilator. Silperisone HCl is used to treat recurrent painful myoclonus due to spinal cord injury, abnormal hypertonia due to cerebrovascular disease, dystonia symptoms, cone tension syndrome, multiple sclerosis myospasm and myelitis. silperisone is a sodium channel protein type 2 alpha channel blocker. silperisone is an organosilicon similar to tolperisone, an organosilicon compound with centrally acting muscle relaxant properties.
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GX-585
GX-585 is a sulfonamide analog that is a Nav 1.7 channel inhibitor with analgesic activity for the study of neuropathic pain and inflammation.
