PNU-282987 is a potent α7 nicotinic acetylcholine receptor (nAChR) agonist with an EC50 of 154 nM. PNU-282987 is also a functional antagonist of the 5-HT3 receptor with an IC50 of 4541 nM. PNU-282987 can be used for the research of central and peripheral nervous systems.

MDH1-IN-2 (Compound 7c) 是一种有效和具有选择性的 MDH1 抑制剂，IC50 为 2.27 μM。MDH1-IN-2 具有研究癌症疾病的潜力。

STF-118804是一种高度特异性的NAMPT抑制剂；降低大多数 B-ALL 细胞系的活力，IC50 <10 nM。