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Lofepramine
CAS No. 23047-25-8
Lofepramine ( Lopramine; Amplit; Leo 640; Gamanil )
产品货号. M26742 CAS No. 23047-25-8
Lofepramine is a potent tricyclic antidepressant that is extensively metabolized to desipramine.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥332 | 有现货 |
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| 5MG | ￥535 | 有现货 |
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| 10MG | ￥737 | 有现货 |
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| 25MG | ￥1523 | 有现货 |
|
| 50MG | ￥2276 | 有现货 |
|
| 100MG | ￥3418 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Lofepramine
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Lofepramine is a potent tricyclic antidepressant that is extensively metabolized to desipramine.
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产品描述Lofepramine is a potent tricyclic antidepressant that is extensively metabolized to desipramine. It inhibits the serotonin and norepinephrine transporters by inhibiting neurons with Kd values of 70 and 5.4 nM, respectively, with weak antagonism of serotonin, histamine and muscarinic receptors.
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同义词Lopramine; Amplit; Leo 640; Gamanil
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体Topo II
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研究领域——
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适应症——
化学信息
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CAS Number23047-25-8
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分子量419.0
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分子式C26H27ClN2O
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纯度>98% (HPLC)
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溶解度——
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SMILESCN(CCCN1c2ccccc2CCc2ccccc12)CC(=O)c1ccc(Cl)cc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.J P Braybrooke, et al. A phase II study of Razoxane, an antiangiogenic topoisomerase II inhibitor, in renal cell cancer with assessment of potential surrogate markers of angiogenesis. Clin Cancer Res.2000; 6(12):4697-704.
产品手册
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