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LP-211

CAS No. 1052147-86-0

LP-211 ( —— )

产品货号. M20108 CAS No. 1052147-86-0

LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥316 有现货
5MG ¥518 有现货
10MG ¥786 有现货
25MG ¥1531 有现货
50MG ¥2608 有现货
100MG ¥4155 有现货
200MG ¥5929 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    LP-211
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.
  • 产品描述
    LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.
  • 同义词
    ——
  • 通路
    Endocrinology/Hormones
  • 靶点
    5-HT Receptor
  • 受体
    5-HT7;D2 receptor;5-HT1A receptor
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1052147-86-0
  • 分子量
    466.62
  • 分子式
    C30H34N4O
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO: 90 mg/mL (192.87 mM)
  • SMILES
    O=C(CCCCCN1CCN(CC1)c1ccccc1-c1ccccc1)NCc1ccc(cc1)C#N
  • 化学全称
    N-[(4-cyanophenyl)methyl]-6-[4-(2-phenylphenyl)piperazin-1-yl]hexanamide

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Leopoldo M et al. Structural modifications of N-(1234-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides: influence on lipophilicity and 5-HT7 receptor activity. Part III. J Med Chem. 2008 Sep 25;51(18):5813-22.
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