LP-211
CAS No. 1052147-86-0
LP-211 ( —— )
产品货号. M20108 CAS No. 1052147-86-0
LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥316 | 有现货 |
|
5MG | ¥518 | 有现货 |
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10MG | ¥786 | 有现货 |
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25MG | ¥1531 | 有现货 |
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50MG | ¥2608 | 有现货 |
|
100MG | ¥4155 | 有现货 |
|
200MG | ¥5929 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称LP-211
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.
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产品描述LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.
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同义词——
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT7;D2 receptor;5-HT1A receptor
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研究领域——
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适应症——
化学信息
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CAS Number1052147-86-0
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分子量466.62
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分子式C30H34N4O
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纯度>98% (HPLC)
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溶解度DMSO: 90 mg/mL (192.87 mM)
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SMILESO=C(CCCCCN1CCN(CC1)c1ccccc1-c1ccccc1)NCc1ccc(cc1)C#N
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化学全称N-[(4-cyanophenyl)methyl]-6-[4-(2-phenylphenyl)piperazin-1-yl]hexanamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Leopoldo M et al. Structural modifications of N-(1234-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides: influence on lipophilicity and 5-HT7 receptor activity. Part III. J Med Chem. 2008 Sep 25;51(18):5813-22.
产品手册
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