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LAQ824

CAS No. 404951-53-7

LAQ824 ( Dacinostat )

产品货号. M14389 CAS No. 404951-53-7

LAQ824 (Dacinostat) is a novel HDAC inhibitor with IC50 of 32 nM and is known to activate the p21 promoter.

纯度: >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥502 有现货
5MG ¥907 有现货
10MG ¥1531 有现货
25MG ¥2746 有现货
50MG ¥4155 有现货
100MG ¥6018 有现货
500MG ¥12312 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    LAQ824
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    LAQ824 (Dacinostat) is a novel HDAC inhibitor with IC50 of 32 nM and is known to activate the p21 promoter.
  • 产品描述
    LAQ824 (Dacinostat) is a novel HDAC inhibitor with IC50 of 32 nM and is known to activate the p21 promoter.
  • 同义词
    Dacinostat
  • 通路
    Cell Cycle/DNA Damage
  • 靶点
    HDAC
  • 受体
    HDAC
  • 研究领域
    Cancer
  • 适应症
    ——

化学信息

  • CAS Number
    404951-53-7
  • 分子量
    379.46
  • 分子式
    C22H25N3O3
  • 纯度
    >98%(HPLC)
  • 溶解度
    DMSO: 76 mg/mL (200.28 mM)
  • SMILES
    O=C(NO)/C=C/C1=CC=C(CN(CCO)CCC2=CNC3=C2C=CC=C3)C=C1
  • 化学全称
    (2E)-N-hydroxy-3-[4-[[(2-hydroxyethyl)[2-(1H-indol-3-yl)ethyl]amino]methyl]phenyl]-2-propenamide

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Atadja P, et al. Y Res, 2004, 64(2), 689-695.
产品手册
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