BRD2492
CAS No. 1821669-43-5
BRD2492 ( BRD 2492 )
产品货号. M12810 CAS No. 1821669-43-5
BRD2492 is a highly potent, selective HDAC1/2 inhibitor (IC50=2/19 nM, respectively).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥7857 | 有现货 |
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50MG | ¥16038 | 有现货 |
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100MG | ¥20250 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称BRD2492
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述BRD2492 is a highly potent, selective HDAC1/2 inhibitor (IC50=2/19 nM, respectively).
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产品描述BRD2492 is a highly potent, selective HDAC1/2 inhibitor (IC50=2/19 nM, respectively) that displays excellent selectivity versus HDAC3 (IC50=2.08 uM, ≥110-fold selectivity) and all other HDAC isoforms, increases caspase-3 activation.
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同义词BRD 2492
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通路Cell Cycle/DNA Damage
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靶点HDAC
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受体HDAC
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研究领域——
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适应症——
化学信息
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CAS Number1821669-43-5
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分子量346.39
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分子式C20H18N4O2
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C(NC1=CC(C2=CC=NC=C2)=CC=C1N)C3=CC=C(NC(C)=O)C=C3
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化学全称4-Acetylamino-N-(2-amino-5-pyridin-4-yl-phenyl)-benzamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Wagner FF, et al. ACS Chem Biol. 2016 Feb 19;11(2):363-74.
产品手册
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