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L-732138

CAS No. 148451-96-1

L-732138 ( —— )

产品货号. M21568 CAS No. 148451-96-1

L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM).

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥356 有现货
5MG ¥583 有现货
10MG ¥988 有现货
25MG ¥1847 有现货
50MG ¥3216 有现货
100MG ¥4771 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    L-732138
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM).
  • 产品描述
    L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM).
  • 同义词
    ——
  • 通路
    GPCR/G Protein
  • 靶点
    Neurokinin Receptor
  • 受体
    NK-1
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    148451-96-1
  • 分子量
    472.38
  • 分子式
    C22H18F6N2O3
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)OCc1cc(cc(c1)C(F)(F)F)C(F)(F)F
  • 化学全称
    [35-Bis(trifluoromethyl)phenyl]methyl (2S)-2-acetamido-3-(1H-indol-3-yl)propanoate

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Mu?oz M et al. The NK-1 Receptor Antagonist L-732138 Induces Apoptosis and Counteracts Substance P-Related Mitogenesis in Human Melanoma Cell Lines. Cancers (Basel). 2010 Apr 20;2(2):611-23.
产品手册
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