Ketanserin

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.

A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C; also has a high affinity antagonist for the H1 receptor (Ki= 2 nM) and α1-adrenergic receptor (Ki=40 nM); an antihypertensive agent.Hypertension Approved

R41468

Endocrinology/Hormones

5-HT Receptor

5-HT2A;5-HT2C(Human);5-HT2C(Rat)

Cardiovascular Disease

Hypertension

74050-98-9

395.43

C22H22FN3O3

>98% (HPLC)

DMSO: 8 mg/mL

O=C(N1CCN2CCC(C(C3=CC=C(F)C=C3)=O)CC2)NC4=C(C=CC=C4)C1=O

2,4(1H,3H)-Quinazolinedione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-

(-20℃)

With Ice Pack

≥ 2 years