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KA2507
CAS No. 1636894-46-6
KA2507 ( —— )
产品货号. M23733 CAS No. 1636894-46-6
KA2507 is a potent and selective HDAC6 inibitor with an IC50 of 2.5nM.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1596 | 有现货 |
|
| 10MG | ￥2568 | 有现货 |
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| 25MG | ￥4334 | 有现货 |
|
| 50MG | ￥6253 | 有现货 |
|
| 100MG | ￥8748 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称KA2507
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述KA2507 is a potent and selective HDAC6 inibitor with an IC50 of 2.5nM.
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产品描述KA2507 is a potent and selective HDAC6 inibitor with an IC50 of 2.5nM.
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同义词——
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通路Cell Cycle/DNA Damage
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靶点HDAC
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受体HDAC6; HDAC8
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研究领域——
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适应症——
化学信息
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CAS Number1636894-46-6
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分子量322.3
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分子式C16H14N6O2
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纯度>98% (HPLC)
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溶解度DMSO : 60 mg/mL (186.15 mM; Need ultrasonic)
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SMILESO=C(NO)C1=CC=C(CN(C2=NC=CN=C2)C3=NC=CN=C3)C=C1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Apostolia M Tsimberidou, et al. Preclinical Development and First-in-Human Study of KA2507, a Selective and Potent Inhibitor of Histone Deacetylase 6, for Patients with Refractory Solid Tumors. Clin Cancer Res. 2021 May 4.
产品手册
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