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HA-155

CAS No. 1229652-22-5

HA-155 ( Autotaxin Inhibitor IV )

产品货号. M23406 CAS No. 1229652-22-5

HA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥502 有现货
5MG ¥1069 有现货
10MG ¥1920 有现货
25MG ¥4601 有现货
50MG ¥5792 有现货
100MG ¥7071 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    HA-155
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    HA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.
  • 产品描述
    HA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.
  • 同义词
    Autotaxin Inhibitor IV
  • 通路
    Angiogenesis
  • 靶点
    PDE
  • 受体
    ATX (autotaxin)
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1229652-22-5
  • 分子量
    463.3
  • 分子式
    C24H19BFNO5S
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO:10 mM
  • SMILES
    B(C1=CC=C(C=C1)COC2=CC=C(C=C2)/C=C\3/C(=O)N(C(=O)S3)CC4=CC=C(C=C4)F)(O)O
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Albers H M H G , Hendrickx L J D , Van Tol R J P , et al. Structure-Based Design of Novel Boronic Acid-Based Inhibitors of Autotaxin[J]. Journal of Medicinal Chemistry, 2011, 54(13):4619-26.
产品手册
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