HA-155
CAS No. 1229652-22-5
HA-155 ( Autotaxin Inhibitor IV )
产品货号. M23406 CAS No. 1229652-22-5
HA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥502 | 有现货 |
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5MG | ¥1069 | 有现货 |
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10MG | ¥1920 | 有现货 |
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25MG | ¥4601 | 有现货 |
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50MG | ¥5792 | 有现货 |
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100MG | ¥7071 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称HA-155
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述HA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.
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产品描述HA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.
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同义词Autotaxin Inhibitor IV
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通路Angiogenesis
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靶点PDE
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受体ATX (autotaxin)
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研究领域——
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适应症——
化学信息
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CAS Number1229652-22-5
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分子量463.3
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分子式C24H19BFNO5S
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纯度>98% (HPLC)
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溶解度DMSO:10 mM
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SMILESB(C1=CC=C(C=C1)COC2=CC=C(C=C2)/C=C\3/C(=O)N(C(=O)S3)CC4=CC=C(C=C4)F)(O)O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Albers H M H G , Hendrickx L J D , Van Tol R J P , et al. Structure-Based Design of Novel Boronic Acid-Based Inhibitors of Autotaxin[J]. Journal of Medicinal Chemistry, 2011, 54(13):4619-26.
产品手册
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