
Galnon
CAS No. 475115-35-6
Galnon ( —— )
产品货号. M22086 CAS No. 475115-35-6
Galnon 是一种甘丙肽受体激动剂,可改善皮质骨组织的内在特性 Galnon 的特点是抑制癫痫发作、减少进食行为、减少阿片戒断的体征,并减轻对部分坐骨神经损伤的热痛觉过敏反应。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥2446 | 有现货 |
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10MG | ¥3669 | 有现货 |
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25MG | ¥6618 | 有现货 |
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100MG | 获取报价 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Galnon
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Galnon 是一种甘丙肽受体激动剂,可改善皮质骨组织的内在特性 Galnon 的特点是抑制癫痫发作、减少进食行为、减少阿片戒断的体征,并减轻对部分坐骨神经损伤的热痛觉过敏反应。
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产品描述Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue propertiesGalnon has been characterized to inhibit seizures, decrease feeding behaviour, diminish physical signs of opiate withdrawal and to alleviate heat-hyperalgesic response to partial sciatic nerve injury[1]. Galnon, a GAL receptor agonist, may enhance osteoclastic bone resorption in OVX rats. Although galnon reduced bone volume, biomechanical testing revealed that bone of galnon-treated animals was mechanically superior per unit area. Taken together, galnon simultaneously improves the intrinsic quality of cortical bone whilst stimulating osteoclastic activity in the OVX rat model.
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体外实验——
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体内实验——
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同义词——
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通路GPCR/G Protein
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靶点Neuropeptide Y Receptor
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受体Galanin receptor
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研究领域——
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适应症——
化学信息
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CAS Number475115-35-6
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分子量678.83
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分子式C40H46N4O6
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纯度>98% (HPLC)
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溶解度——
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SMILESCc1cc(=O)oc2cc(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC3CCCCC3)NC(=O)OCC3c4ccccc4-c4ccccc34)ccc12
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献




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Galanin Receptor Lig...
The chimeric peptide M35 [galanin (1-13)-bradykinin(2-9) amide] is a high-affinity galanin receptor ligand acting as a galanin receptor antagonist in the rat spinal cord, rat hippocampus and isolated mouse pancreatic islets. The radiolabelled M35 and performed equilibrium binding studies with [125I] M35 on the rat pancreatic beta-cell line Rin m 5F.
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CART (55-102) (rat)
Cocaine- and amphetamine-regulated transcript (CART) with potent appetite-suppressing activity. Satiety factor; inhibits normal and starvation-induced feeding. Closely related to the actions of leptin and neuropeptide Y; blocks the neuropeptide Y-induced feeding response. Induces anxiety and stress behavior in rodents.
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Velneperit
Velneperit 是一种有效的选择性神经肽 Y (NPY) Y5 受体,正在评估其治疗肥胖的效果。