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Galnon

CAS No. 475115-35-6

Galnon ( —— )

产品货号. M22086 CAS No. 475115-35-6

Galnon 是一种甘丙肽受体激动剂,可改善皮质骨组织的内在特性 Galnon 的特点是抑制癫痫发作、减少进食行为、减少阿片戒断的体征,并减轻对部分坐骨神经损伤的热痛觉过敏反应。

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥2446 有现货
10MG ¥3669 有现货
25MG ¥6618 有现货
100MG 获取报价 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Galnon
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Galnon 是一种甘丙肽受体激动剂,可改善皮质骨组织的内在特性 Galnon 的特点是抑制癫痫发作、减少进食行为、减少阿片戒断的体征,并减轻对部分坐骨神经损伤的热痛觉过敏反应。
  • 产品描述
    Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue propertiesGalnon has been characterized to inhibit seizures, decrease feeding behaviour, diminish physical signs of opiate withdrawal and to alleviate heat-hyperalgesic response to partial sciatic nerve injury[1]. Galnon, a GAL receptor agonist, may enhance osteoclastic bone resorption in OVX rats. Although galnon reduced bone volume, biomechanical testing revealed that bone of galnon-treated animals was mechanically superior per unit area. Taken together, galnon simultaneously improves the intrinsic quality of cortical bone whilst stimulating osteoclastic activity in the OVX rat model.
  • 体外实验
    ——
  • 体内实验
    ——
  • 同义词
    ——
  • 通路
    GPCR/G Protein
  • 靶点
    Neuropeptide Y Receptor
  • 受体
    Galanin receptor
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    475115-35-6
  • 分子量
    678.83
  • 分子式
    C40H46N4O6
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    Cc1cc(=O)oc2cc(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC3CCCCC3)NC(=O)OCC3c4ccccc4-c4ccccc34)ccc12
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Sollenberg U , Bartfai T , Langel U . Galnon - A low-molecular weight ligand of the galanin receptors[J]. Neuropeptides, 2005, 39(3):161-163.
产品手册
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