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Velneperit
CAS No. 342577-38-2
Velneperit ( S2367 )
产品货号. M22270 CAS No. 342577-38-2
Velneperit 是一种有效的选择性神经肽 Y (NPY) Y5 受体，正在评估其治疗肥胖的效果。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥356 | 有现货 |
|
| 5MG | ￥583 | 有现货 |
|
| 10MG | ￥988 | 有现货 |
|
| 25MG | ￥2203 | 有现货 |
|
| 50MG | ￥3750 | 有现货 |
|
| 100MG | ￥5524 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Velneperit
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Velneperit 是一种有效的选择性神经肽 Y (NPY) Y5 受体，正在评估其治疗肥胖的效果。
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产品描述Velneperit is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.
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体外实验——
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体内实验——
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同义词S2367
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通路GPCR/G Protein
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靶点Neuropeptide Y Receptor
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受体neuropeptide Y (NPY) Y5 receptor
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研究领域Others
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适应症Obesity
化学信息
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CAS Number342577-38-2
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分子量407.45
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分子式C17H24F3N3O3S
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纯度>98% (HPLC)
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溶解度DMSO:29 mg/mL (71.17 mM)
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SMILESFC(F)(F)C1=CN=C(NC([C@H]2CC[C@H](NS(=O)(C(C)(C)C)=O)CC2)=O)C=C1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
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M871
Selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM for GAL2 and GAL1 receptors respectively). Blocks the pro-nociceptive effect of GAL2 receptor agonists.
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M 1145
Potent and selective galanin receptor 2 (GAL2) agonist (EC50 = 38 nM, Ki values are 6.55, 497 and 587 nM at GAL2, GAL3 and GAL1 respectively). Has an additive effect on the signal transduction of galanin.
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[D-Trp34]-Neuropepti...
Potent neuropeptide Y (NPY) Y5 receptor agonist (pEC50 values are 7.82, 6.28, 6.44 and > 6 at rat Y5, Y4, Y1 and Y2 receptors respectively) that displays > 26-fold, > 1000-fold and > 1000-fold selectivity over Y1, Y2 and Y4 receptors respectively. Induces hyperphagia, body weight gain, adiposity, hypercholesterolemia, hyperinsulinemia and hyperleptinemia in vivo. Orally active.
