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GSK-4716

CAS No. 101574-65-6

GSK-4716 ( —— )

产品货号. M20159 CAS No. 101574-65-6

GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥308 有现货
10MG ¥470 有现货
25MG ¥1061 有现货
50MG ¥2041 有现货
100MG ¥3799 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    GSK-4716
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.
  • 产品描述
    GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.
  • 同义词
    ——
  • 通路
    Endocrinology/Hormones
  • 靶点
    Estrogen Receptor/ERR
  • 受体
    ERRβ/γ
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    101574-65-6
  • 分子量
    282.34
  • 分子式
    C17H18N2O2
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO:100 mg/mL?(354.18 mM)
  • SMILES
    CC(C)c1ccc(cc1)\C=N\NC(=O)c1ccc(O)cc1
  • 化学全称
    4-hydroxy-N-[(4-propan-2-ylphenyl)methylideneamino]benzamide

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Wang L Zuercher W J Consler T G et al. X-ray Crystal Structures of the Estrogen-related Receptor- Ligand Binding Domain in Three Functional States Reveal the Molecular Basis of Small Molecule Regulation[J]. Journal of Biological Chemistry 2006 281(49):37773-37781.
产品手册
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