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GSK-4716
CAS No. 101574-65-6
GSK-4716 ( —— )
产品货号. M20159 CAS No. 101574-65-6
GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥308 | 有现货 |
|
| 10MG | ￥470 | 有现货 |
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| 25MG | ￥1061 | 有现货 |
|
| 50MG | ￥2041 | 有现货 |
|
| 100MG | ￥3799 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称GSK-4716
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.
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产品描述GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.
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同义词——
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通路Endocrinology/Hormones
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靶点Estrogen Receptor/ERR
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受体ERRβ/γ
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研究领域——
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适应症——
化学信息
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CAS Number101574-65-6
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分子量282.34
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分子式C17H18N2O2
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纯度>98% (HPLC)
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溶解度DMSO:100 mg/mL?(354.18 mM)
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SMILESCC(C)c1ccc(cc1)\C=N\NC(=O)c1ccc(O)cc1
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化学全称4-hydroxy-N-[(4-propan-2-ylphenyl)methylideneamino]benzamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Wang L Zuercher W J Consler T G et al. X-ray Crystal Structures of the Estrogen-related Receptor- Ligand Binding Domain in Three Functional States Reveal the Molecular Basis of Small Molecule Regulation[J]. Journal of Biological Chemistry 2006 281(49):37773-37781.
产品手册
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