GSK-25
CAS No. 874119-56-9
GSK-25 ( —— )
产品货号. M17637 CAS No. 874119-56-9
GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and p70S6K (RSK1 IC50 of 398 nM, p70S6K IC50 of 1000nM), and a dramatically improved P450 profile (>2.2 uM at all isozymes tested).
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥437 | 有现货 |
|
5MG | ¥680 | 有现货 |
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10MG | ¥964 | 有现货 |
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25MG | ¥1458 | 有现货 |
|
50MG | ¥2317 | 有现货 |
|
100MG | ¥3872 | 有现货 |
|
200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称GSK-25
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and p70S6K (RSK1 IC50 of 398 nM, p70S6K IC50 of 1000nM), and a dramatically improved P450 profile (>2.2 uM at all isozymes tested).
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产品描述GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and p70S6K (RSK1 IC50 of 398 nM, p70S6K IC50 of 1000nM), and a dramatically improved P450 profile (>2.2 uM at all isozymes tested).
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同义词——
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通路Others
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靶点Other Targets
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受体RSK1; mTOR (p70S6K)
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研究领域——
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适应症——
化学信息
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CAS Number874119-56-9
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分子量513.34
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分子式C24H16Cl2F2N6O
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纯度98%
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溶解度——
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SMILESClc1nccc(c1)C=2NC(C)=C(C(N=2)c3ccc(Cl)cc3F)C(=O)Nc4cc5cnnc5cc4F
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Sehon CA, et al. J Med Chem. 2008 Nov 13;51(21):6631-4.
产品手册
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