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GR-64349

CAS No. 137593-52-3

GR-64349 ( GR64349 )

产品货号. M11556 CAS No. 137593-52-3

GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
100MG 获取报价 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    GR-64349
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM.
  • 产品描述
    GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM, displays >1000- and >300-fold selectivity over NK1 and NK3 receptors, respectively.Pain Discontinued
  • 同义词
    GR64349
  • 通路
    GPCR/G Protein
  • 靶点
    Neurokinin Receptor
  • 受体
    Neurokinin Receptor
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    137593-52-3
  • 分子量
    921.12
  • 分子式
    C42H68N10O11S
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    CC(C)CC(C(=O)NC(CCSC)C(=O)N)N1CCC(C1=O)NC(=O)C(C(C)C)NC(=O)C(CC2=CC=CC=C2)NC(=O)C(CO)NC(=O)C(CC(=O)O)NC(=O)C(CCCCN)N
  • 化学全称
    KDSFVGLM (Modifications: Leu-7 = R-γ-lactam-Leu, Met-8 = C-terminal amide)

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Deal MJ, et al. J Med Chem. 1992 Oct 30;35(22):4195-204.
2. Chizh BA, et al. Br J Pharmacol. 1995 Jul;115(6):1013-9.
3. Chang Y, et al. J Pharmacol Exp Ther. 2000 Jul;294(1):147-54.
产品手册
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