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GR-64349
CAS No. 137593-52-3
GR-64349 ( GR64349 )
产品货号. M11556 CAS No. 137593-52-3
GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 100MG | 获取报价 | 有现货 |
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| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称GR-64349
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM.
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产品描述GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM, displays >1000- and >300-fold selectivity over NK1 and NK3 receptors, respectively.Pain Discontinued
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同义词GR64349
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通路GPCR/G Protein
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靶点Neurokinin Receptor
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受体Neurokinin Receptor
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研究领域——
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适应症——
化学信息
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CAS Number137593-52-3
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分子量921.12
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分子式C42H68N10O11S
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纯度>98% (HPLC)
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溶解度——
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SMILESCC(C)CC(C(=O)NC(CCSC)C(=O)N)N1CCC(C1=O)NC(=O)C(C(C)C)NC(=O)C(CC2=CC=CC=C2)NC(=O)C(CO)NC(=O)C(CC(=O)O)NC(=O)C(CCCCN)N
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化学全称KDSFVGLM (Modifications: Leu-7 = R-γ-lactam-Leu, Met-8 = C-terminal amide)
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Deal MJ, et al. J Med Chem. 1992 Oct 30;35(22):4195-204.
2. Chizh BA, et al. Br J Pharmacol. 1995 Jul;115(6):1013-9.
3. Chang Y, et al. J Pharmacol Exp Ther. 2000 Jul;294(1):147-54.
2. Chizh BA, et al. Br J Pharmacol. 1995 Jul;115(6):1013-9.
3. Chang Y, et al. J Pharmacol Exp Ther. 2000 Jul;294(1):147-54.
产品手册
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