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Filaminast

CAS No. 141184-34-1

Filaminast ( WAY-PDA-641;PDA-641;WAY-123641 )

产品货号. M11714 CAS No. 141184-34-1

Filaminast (WAY-PDA-641;PDA-641;WAY-123641) is a potent and selective PDE4 inhibitor with IC50 of 420 nM, displays 36-fold selectivity over PDE3.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥7857 有现货
10MG ¥10449 有现货
25MG ¥15795 有现货
50MG ¥21222 有现货
100MG ¥28593 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Filaminast
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Filaminast (WAY-PDA-641;PDA-641;WAY-123641) is a potent and selective PDE4 inhibitor with IC50 of 420 nM, displays 36-fold selectivity over PDE3.
  • 产品描述
    Filaminast (WAY-PDA-641;PDA-641;WAY-123641) is a potent and selective PDE4 inhibitor with IC50 of 420 nM, displays 36-fold selectivity over PDE3; significantly potentiates the relaxant effects of albuterol, reverses tracheal contractions induced by prostaglandin F2 alpha, leukotriene D4 or histamine in a biphasic manner.Asthma Phase 2 Discontinued
  • 同义词
    WAY-PDA-641;PDA-641;WAY-123641
  • 通路
    Angiogenesis
  • 靶点
    PDE
  • 受体
    PDE
  • 研究领域
    Inflammation/Immunology
  • 适应症
    Asthma

化学信息

  • CAS Number
    141184-34-1
  • 分子量
    292.34
  • 分子式
    C15H20N2O4
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    C(\C)(=N/OC(=O)N)c1cc(c(cc1)OC)OC1CCCC1
  • 化学全称
    1-(3-(Cyclopentyloxy)-4-methoxyphenyl)ethanone-(E)-O-(aminocarbonyl)oxime

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Heaslip RJ, et al. J Pharmacol Exp Ther. 1994 Feb;268(2):888-96.
产品手册
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