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Elevenostat

CAS No. 1454902-97-6

Elevenostat ( JB3-22 )

产品货号. M28876 CAS No. 1454902-97-6

Elevenostat is an HDAC11-selective inhibitor with an IC50 value of 0.235?μM.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥316 有现货
10MG ¥518 有现货
25MG ¥988 有现货
50MG ¥1596 有现货
100MG ¥2973 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Elevenostat
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Elevenostat is an HDAC11-selective inhibitor with an IC50 value of 0.235?μM.
  • 产品描述
    Elevenostat is an HDAC11-selective inhibitor with an IC50 value of 0.235?μM.(In Vitro):Elevenostat induced cell death in MM cell lines.(In Vivo):Elevenostat produced similar anti-MM activity in vivo, improving survival among mice inoculated with 5TGM1 MM cells.
  • 同义词
    JB3-22
  • 通路
    Cell Cycle/DNA Damage
  • 靶点
    HDAC
  • 受体
    Telomerase
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1454902-97-6
  • 分子量
    315.3
  • 分子式
    C16H17N3O4
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    COc(cccc1)c1NC(NCc(cc1)ccc1C(NO)=O)=O
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Fleming AM, et al. Human DNA Repair Genes Possess Potential G-Quadruplex Sequences in Their Promoters and 5'-Untranslated Regions. Biochemistry. 2018 Feb 13;57(6):991-1002.
产品手册
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