Eletriptan ( UK 116044 )

产品货号. M11842 CAS No. 143322-58-1

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.

纯度: >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

规格	价格/人民币	库存	数量
50MG	￥15317	有现货
100MG	获取报价	有现货
200MG	获取报价	有现货
500MG	获取报价	有现货
1G	获取报价	有现货

拼团产品询价大包装询价加入购物车

生物学信息

产品名称

Eletriptan
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.
产品描述

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist; significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease; displays antimigraine activity.Migraine Approved
同义词

UK 116044
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT Receptor
研究领域

Neurological Disease
适应症

Migraine

化学信息

CAS Number

143322-58-1
分子量

382.52
分子式

C22H26N2O2S
纯度

>98% (HPLC)
溶解度

——
SMILES

CN1CCC[C@@H]1Cc2c[nH]c3c2cc(cc3)CCS(=O)(=O)c4ccccc4
化学全称

3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole

运输与储存

储存条件

(-20℃)
运输条件

With Ice Pack
稳定性

≥ 2 years

参考文献

1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.
2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.
3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.

计算器

浓度计算器

摩尔计算器

分子量计算器

产品手册

关联产品

Donitriptan hydrochl...

Donitriptan hydrochloride is a potent, high efficacy agonist of 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectively.
LP-211

LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.
Loxapine succinate

A typical antipsychotic agent that displays an extremely strong binding affinity for dopamine D4 and serotonin 5-HT2 receptors.

Product			Quantity Required*
Name *			E-mail Address *
Organization *			Phone Number
Remarks