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Droloxifene
CAS No. 82413-20-5
Droloxifene ( 3-Hydroxytamoxifen;FK-435 )
产品货号. M16060 CAS No. 82413-20-5
A nonsteroidal selective estrogen receptor modulator (SERM) that shows 10- to 60-fold increased affinity for the estrogen receptor compared with Tamoxifen.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1596 | 有现货 |
|
| 10MG | ￥2406 | 有现货 |
|
| 25MG | ￥4180 | 有现货 |
|
| 50MG | ￥5962 | 有现货 |
|
| 100MG | ￥7995 | 有现货 |
|
| 500MG | ￥16038 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Droloxifene
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述A nonsteroidal selective estrogen receptor modulator (SERM) that shows 10- to 60-fold increased affinity for the estrogen receptor compared with Tamoxifen.
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产品描述A nonsteroidal selective estrogen receptor modulator (SERM) that shows 10- to 60-fold increased affinity for the estrogen receptor compared with Tamoxifen; has reduced partial estrogen agonistic activity.Breast Cancer Phase 2 Clinical
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同义词3-Hydroxytamoxifen;FK-435
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通路Endocrinology/Hormones
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靶点Estrogen Receptor/ERR
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受体Estrogen Receptor/ERR
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研究领域Cancer
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适应症Breast Cancer
化学信息
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CAS Number82413-20-5
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分子量387.52
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分子式C26H29NO2
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纯度>98% (HPLC)
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溶解度——
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SMILESCCC(=C(C1=CC=C(C=C1)OCCN(C)C)C2=CC(=CC=C2)O)C3=CC=CC=C3
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化学全称(Z)-4-(1-(4-(2-aminoethoxy)phenyl)-2-phenylbut-1-en-1-yl)phenol
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Rauschning W, et al. Breast Cancer Res Treat. 1994;31(1):83-94.
2. Hasmann M, et al. Cancer Lett. 1994 Sep 15;84(2):101-16.
3. Leng Y, et al. Eur J Pharmacol. 2000 Dec 8;409(2):123-31.
2. Hasmann M, et al. Cancer Lett. 1994 Sep 15;84(2):101-16.
3. Leng Y, et al. Eur J Pharmacol. 2000 Dec 8;409(2):123-31.
产品手册
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