Deriglidole ( —— )

产品货号. M32880 CAS No. 122830-14-2

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Deriglidole
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Deriglidole 是外周肾上腺素能受体拮抗剂，对 α2 肾上腺素受体具有高亲和力。
产品描述

Deriglidole is a peripheral adrenoceptor antagonist with a high affinity for α2-adrenoceptors.
体外实验

Deriglidole is a selective α2-receptor inhibitor. Deriglidole inhibits [3H]Clonidine and [3H]Idazoxan but not [3H]Prazosin binding to rat cortical and human platelet α2-adrenoceptors and is more selective than Idazoxan for peripheral receptors.
体内实验

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同义词

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通路

GPCR/G Protein
靶点

Adrenergic Receptor
受体

Adrenergic Receptor
研究领域

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适应症

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1. Natali A,et al. Effects of acute alpha 2-blockade on insulin action and secretion in humans. Am J Physiol. 1998 Jan;274(1 Pt 1):E57-64.?

计算器

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