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Cerlapirdine
CAS No. 925448-93-7
Cerlapirdine ( SAM531; SAM-531; SAM 531; PF-05212365; P -05212365; WAY-262,531 )
产品货号. M27966 CAS No. 925448-93-7
Cerlapirdine is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1442 | 有现货 |
|
| 10MG | ￥2341 | 有现货 |
|
| 25MG | ￥4633 | 有现货 |
|
| 50MG | ￥6658 | 有现货 |
|
| 100MG | ￥9153 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Cerlapirdine
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Cerlapirdine is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
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产品描述Cerlapirdine is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
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同义词SAM531; SAM-531; SAM 531; PF-05212365; P -05212365; WAY-262,531
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体hSmo;mSmo
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研究领域——
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适应症——
化学信息
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CAS Number925448-93-7
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分子量409.5
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分子式C22H23N3O3S
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纯度>98% (HPLC)
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溶解度——
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SMILESCN(C)CCCOc1ccc2n[nH]c(c2c1)S(=O)(=O)c1cccc2ccccc12
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Lauressergues E, et al. Pharmacological evaluation of a series of smoothened antagonists in signaling pathways and after topical application in a depilated mouse model. Pharmacol Res Perspect. 2016 Mar 4;4(2):e00214.
产品手册
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