Canertinib
CAS No. 267243-28-7
Canertinib ( CI-1033; PD-183805 )
产品货号. M18334 CAS No. 267243-28-7
Canertinib is a pan-erbB tyrosine kinase inhibitor which work against esophageal squamous cell carcinoma in vitro and in vivo.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥251 | 有现货 |
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10MG | ¥405 | 有现货 |
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25MG | ¥518 | 有现货 |
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50MG | ¥640 | 有现货 |
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100MG | 获取报价 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Canertinib
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Canertinib is a pan-erbB tyrosine kinase inhibitor which work against esophageal squamous cell carcinoma in vitro and in vivo.
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产品描述Canertinib is a pan-erbB tyrosine kinase inhibitor which work against esophageal squamous cell carcinoma in vitro and in vivo. Canertinib treatment significantly affects tumour metabolism, proliferation and hypoxia as determined by PET.
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同义词CI-1033; PD-183805
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通路Others
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靶点Other Targets
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受体EGFR; HER2/ErbB2
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研究领域Cancer
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适应症——
化学信息
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CAS Number267243-28-7
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分子量485.94
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分子式C24H25ClFN5O3
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纯度98%
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溶解度DMSO : 4.9 mg/mL 10.08 mM;
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SMILESC=CC(=O)Nc1c(cc2c(c1)c(ncn2)Nc1cc(c(cc1)F)Cl)OCCCN1CCOCC1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Smaill JB et al. J Med Chem. 2000; 43(7): 1380-1397.
产品手册
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