Bilastine
CAS No. 202189-78-4
Bilastine ( Bilastine trade name Bilaxten )
产品货号. M18206 CAS No. 202189-78-4
Bilastine is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of action.
纯度: 98%
规格 | 价格/人民币 | 库存 | 数量 |
25MG | ¥316 | 有现货 |
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50MG | ¥518 | 有现货 |
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100MG | ¥851 | 有现货 |
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200MG | ¥1256 | 有现货 |
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500MG | ¥2122 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Bilastine
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Bilastine is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of action.
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产品描述Bilastine (trade name Bilaxten) is a second generation antihistamine drug for the treatment of allergic rhinoconjunctivitis and urticaria (hives). It exerts its effect as a selective histamine H1 receptor antagonist, and has a potency similar to cetirizine and is superior to fexofenadine. It was developed in Spain by FAES Farma. Bilastine is approved in the European Union for the symptomatic treatment of allergic rhinoconjunctivitis and urticaria, but it is not approved by the U.S. Food and Drug Administration for any use in the United States. Bilastine has been effective in the treatment of ocular symptoms and diseases of allergies, including rhinoconjuctivitis. Additionally, bilastine has been shown to improve quality of life, and all nasal and ocular symptoms related to allergic rhinitis.
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同义词Bilastine trade name Bilaxten
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体H1 receptor
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研究领域Inflammation/Immunology
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适应症——
化学信息
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CAS Number202189-78-4
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分子量463.62
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分子式C28H37N3O3
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纯度98%
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溶解度DMSO : ≥ 49.3 mg/mL; 106.34 mM
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SMILESCCOCCn1c(nc2ccccc12)C1CCN(CCc2ccc(cc2)C(C)(C)C(O)=O)CC1
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化学全称2-(4-(2-(4-(1-(2-ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoic acid
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
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Cinitapride
Cinitapride is a gastroprokinetic agent. It slows the actions of the muscles to reduce the symptoms of conditions such as acid reflux, delayed gastric emptying, and ulcer dyspepsia.
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Nafronyl oxalate
A drug used in the management of peripheral and cerebral vascular disorders. It is claimed to enhance cellular oxidative capacity and to be a spasmolytic.
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Homoeriodictyol
Homoeriodictyol, a naturally occurring, bitter-masking flavanone, as a promising agent to increase appetite and food intake. The flavanone homoeriodictyol can increase SGLT-1-mediated glucose uptake but decrease serotonin release in differentiated Caco-2 cells.In contrast to other polyphenols, the flavanon Homoeriodictyol promotes glucose uptake by 29.0 ± 3.83% at a concentration of 100 μM.