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BRD-IN-26
CAS No. 1915012-19-9
BRD-IN-26 ( —— )
产品货号. M13002 CAS No. 1915012-19-9
BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM.
纯度: >98% (HPLC)
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规格 | 价格/人民币 | 库存 | 数量 |
100MG | 获取报价 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称BRD-IN-26
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM.
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产品描述BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM, SMARCA2B and SMARCA4 with KD values of 262 and 417 nM, respectively; displays excellent selectivity over other bromodomains.
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同义词——
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通路Chromatin/Epigenetic
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靶点Bromodomain
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受体Bromodomain
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研究领域——
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适应症——
化学信息
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CAS Number1915012-19-9
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分子量330.82
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分子式C17H19ClN4O
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纯度>98% (HPLC)
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溶解度——
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SMILES——
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化学全称(E)-6-chloro-3-((4-methylpiperazin-1-yl)methylene)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-one
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Sutherell CL, et al. J Med Chem. 2016 May 26;59(10):5095-101.
产品手册
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