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Azalanstat

CAS No. 143393-27-5

Azalanstat ( —— )

产品货号. M34054 CAS No. 143393-27-5

Azalanstat (RS 21607) is an orally available selective mammalian lanosterol 14-alpha-demethylase inhibitor with hypocholesterolemic activity that inhibits cholesterol synthesis in HepG2 cells, human fibroblasts, hamster hepatocytes, and hamster livers through inhibition of the cytochrome P450 enzyme, lanosterol 14 alpha demethylase.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
25MG ¥11886 有现货
50MG ¥15484 有现货
100MG ¥19125 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Azalanstat
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Azalanstat (RS 21607) is an orally available selective mammalian lanosterol 14-alpha-demethylase inhibitor with hypocholesterolemic activity that inhibits cholesterol synthesis in HepG2 cells, human fibroblasts, hamster hepatocytes, and hamster livers through inhibition of the cytochrome P450 enzyme, lanosterol 14 alpha demethylase.
  • 产品描述
    Azalanstat (RS 21607) is an orally available selective mammalian lanosterol 14-alpha-demethylase inhibitor with hypocholesterolemic activity that inhibits cholesterol synthesis in HepG2 cells, human fibroblasts, hamster hepatocytes, and hamster livers through inhibition of the cytochrome P450 enzyme, lanosterol 14 alpha demethylase.
  • 体外实验
    ——
  • 体内实验
    ——
  • 同义词
    ——
  • 通路
    Metabolic Enzyme/Protease
  • 靶点
    P450
  • 受体
    P450
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    143393-27-5
  • 分子量
    429.96
  • 分子式
    C22H24ClN3O2S
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    C([C@]1(CCC2=CC=C(Cl)C=C2)O[C@H](CSC3=CC=C(N)C=C3)CO1)N4C=CN=C4
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

产品手册
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