Atogepant ( MK-8031;AGN-241689 )

产品货号. M11545 CAS No. 1374248-81-3

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Atogepant
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

A potent, selective and orally available CGRP receptor antagonist for the prevention of migraine.
产品描述

A potent, selective and orally available CGRP receptor antagonist for the prevention of migraine.Migraine Phase 3 Clinical
同义词

MK-8031;AGN-241689
通路

GPCR/G Protein
靶点

CGRP Receptor
受体

CGRP Receptor
研究领域

Neurological Disease
适应症

Migraine

CAS Number

1374248-81-3
分子量

603.53
分子式

C29H23F6N5O3
纯度

>98% (HPLC)
溶解度

10 mM in DMSO
SMILES

O=C(C1=CN=C2C(C[C@@]3(C4=CC=CN=C4NC3=O)C2)=C1)N[C@@H]5C(N(CC(F)(F)F)[C@H](C)[C@H](C6=C(F)C=CC(F)=C6F)C5)=O
化学全称

(3'S)-N-[(3S,5S,6R)-6-methyl-2-oxo-1-(2,2,2-trifluoroethyl)-5-(2,3,6-trifluorophenyl)piperidin-3-yl]-2'-oxo-1',2',5,7-tetrahydrospiro[cyclopenta[b]pyridine-6,3'-pyrrolo[2,3-b]pyridine]-3-carboxamide

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