(R)-(-)-Rolipram
CAS No. 85416-75-7
(R)-(-)-Rolipram ( R)-Rolipram;(-)-Rolipram )
产品货号. M16203 CAS No. 85416-75-7
A more active enantiomer of the PDE4 inhibitor rolipram.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥316 | 有现货 |
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5MG | ¥502 | 有现货 |
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10MG | ¥794 | 有现货 |
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25MG | ¥1531 | 有现货 |
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50MG | ¥2851 | 有现货 |
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100MG | 获取报价 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称(R)-(-)-Rolipram
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述A more active enantiomer of the PDE4 inhibitor rolipram.
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产品描述A more active enantiomer of the PDE4 inhibitor rolipram; shows 2-10-fold more potent than the S-(+) enantiomer rolipram.Asthma Phase 2 Clinical
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同义词R)-Rolipram;(-)-Rolipram
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通路Angiogenesis
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靶点PDE
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受体PDE
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研究领域Inflammation/Immunology
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适应症Asthma
化学信息
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CAS Number85416-75-7
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分子量275.34
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分子式C16H21NO3
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纯度>98% (HPLC)
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溶解度DMSO: ≥ 49 mg/mL
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SMILESCOC1=C(C=C(C=C1)C2CC(=O)NC2)OC3CCCC3
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化学全称2-Pyrrolidinone, 4-[3-(cyclopentyloxy)-4-methoxyphenyl]-, (4R)-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Schneider HH, et al. Eur J Pharmacol. 1986 Aug 7;127(1-2):105-15.
2. Owens RJ, et al. Biochem J. 1997 Aug 15;326 ( Pt 1):53-60.
3. Ohsawa F, et al. Jpn J Pharmacol. 1998 Jun;77(2):147-54.
2. Owens RJ, et al. Biochem J. 1997 Aug 15;326 ( Pt 1):53-60.
3. Ohsawa F, et al. Jpn J Pharmacol. 1998 Jun;77(2):147-54.
产品手册
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