UUN44923 ( FTO-IN-1 )

产品货号. M24020 CAS No. 2243944-92-3

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

UUN44923
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

UUN44923 是一种 FTO 抑制剂。它可能有助于治疗相关疾病。 FTO的目标包括肥胖、代谢综合征(MS)、2型糖尿病(T2D)、阿尔茨海默病、乳腺癌、小细胞肺癌、人骨髓横纹肌癌、胰腺癌、恶性胶质母细胞瘤等。
产品描述

UUN44923 is a FTO inhibitor.?It may be useful for treating diseases assocd.?with FTO targets, obesity, metabolic syndrome (MS) , type 2 diabetes (T2D) , Alzheimer's diseases, breast cancers, small- cell lung cancers, a human bone marrow striated muscle cancer, a pancreatic cancer, malignant glioblastoma and the like.?
体外实验

FTO-IN-1 (50 μM) inhibits FTO enzyme activity by 62% in vitro.FTO-IN-1 (50 μM) inhibits the viability of SCLC-21H, RH30 and KP3 cells, with IC50s of 2.1 μM, 5.3 μM, and 5.6 μM, respectively.
体内实验

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同义词

FTO-IN-1
通路

Others
靶点

Other Targets
受体

FTO
研究领域

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适应症

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计算器

产品手册

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