Picloxydine has antiplaque and antibacterial activity. Picloxydine has a destructive effect on the bacterial cell wall and plasma membrane, which leads to cell lysis and release of intracellular components.

Deacylketoconazole is a Ketoconazole derivative and is also an antifungal agent.

DuP-721 is a broad spectrum and orally active antibacterial agent against a variety of clinically susceptible and resistant bacteria, especially M. tuberculosis.