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Tradipitant
CAS No. 622370-35-8
Tradipitant ( VLY-686; LY686017 )
产品货号. M26851 CAS No. 622370-35-8
Tradipitant is an antagonist of neurokinin-1.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥624 | 有现货 |
|
| 5MG | ￥988 | 有现货 |
|
| 10MG | ￥1596 | 有现货 |
|
| 25MG | ￥2811 | 有现货 |
|
| 50MG | ￥4180 | 有现货 |
|
| 100MG | ￥5962 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Tradipitant
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Tradipitant is an antagonist of neurokinin-1.
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产品描述Tradipitant is an antagonist of neurokinin-1.(In Vitro):Tradipitant binds to sections of guinea pig brain with a distribution similar to that previously reported for NK-1 receptors. Areas with the highest density are the accessory olfactory nucleus, anteroventral thalamic nucleus, paraventricular hypothalamic nucleus central amygdaloid nucleus (lateral), and the medial amygdaloid nucleus .(In Vivo):Tradipitant (intravenously administered) treatment localizes in the guinea pig brain and has a distribution similar to that described for the NK-1 receptor using agonist or antagonist radioligands .
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同义词VLY-686; LY686017
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通路GPCR/G Protein
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靶点Neurokinin Receptor
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受体Nucleoside Antimetabolite/Analog
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研究领域——
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适应症——
化学信息
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CAS Number622370-35-8
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分子量587.9
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分子式C28H16ClF6N5O
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纯度>98% (HPLC)
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溶解度——
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SMILESFC(F)(F)c1cc(Cn2nnc(c2-c2ccncc2)-c2ncccc2C(=O)c2ccccc2Cl)cc(c1)C(F)(F)F
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Raynal NJ, et al. 3-Deazauridine enhances the antileukemic action of 5-aza-2'-deoxycytidine and targets drug-resistance due to deficiency in deoxycytidine kinase. Leuk Res. 2011 Jan;35(1):110-8.
产品手册
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