Tirasemtiv

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

Tirasemtiv(CK 2017357) is a small-molecule fast-skeletal-troponin activator, with a potential treatment for muscle weakness and neuromuscular dysfunction.

Tirasemtiv, also known as CK2017357, is a novel skeletal muscle activator. Tirasemtiv slows the rate of calcium release from troponin, thus sensitizing fast skeletal muscle fibers to calcium. Tirasemtiv demonstrated increases in skeletal muscle force in response to neuronal input and delays in the onset and reductions in the degree of muscle fatigue.

CK2017357; CK-2017357; CK 2017357; Tirasemtiv

Others

Other Targets

Troponin

Neurological Disease

——

1005491-05-3

230.27

C12H14N4O

98%

DMSO : ≥ 52 mg/mL 225.82 mM

CCC(CC)n1c2nc(cnc2[nH]c1=O)C#C

1-(1-Ethylpropyl)-6-ethynyl-1,3-dihydro-2H-imidazo(4,5-b)pyrazin-2-one

(-20℃)

With Ice Pack

≥ 2 years