Tenatoprazole ( TU-199; Tenatoprazole; Ulsacare; Protop )

产品货号. M17835 CAS No. 113712-98-4

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Tenatoprazole
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Tenatoprazole, a prodrug of the proton pump inhibitor (PPI) class, can inhibit proton transport (IC50: 3.2 μM).
产品描述

Tenatoprazole, also known as TU-199, is a proton pump inhibitor drug candidate that was undergoing clinical testing as a potential treatment for reflux oesophagitis and peptic ulcer. Tenatoprazole has an imidazopyridine ring in place of the benzimidazole moiety found in other proton pump inhibitors, and has a half-life about seven times longer than other PPIs.
同义词

TU-199; Tenatoprazole; Ulsacare; Protop
通路

Others
靶点

Other Targets
受体

Proton pump
研究领域

Inflammation/Immunology
适应症

——

CAS Number

113712-98-4
分子量

346.4
分子式

C16H18N4O3S
纯度

98%
溶解度

——
SMILES

COc1ccc2[nH]c(nc2n1)S(=O)Cc1c(C)c(OC)c(C)cn1
化学全称

5-methoxy-2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methylsulfinyl]-1H-imidazo[4,5-b]pyridine

1. Shin JM, et al. Biochem Pharmacol, 2006, 71(6), 837-849.

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