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THIP

CAS No. 64603-91-4

THIP ( Gaboxadol; Gaboxadolum )

产品货号. M26482 CAS No. 64603-91-4

THIP has a strong affinity for the δ subunit of GABAA receptors. THIP is a functionally selective GABAAR ligand, agonistic to α4β1δ, α4β3δ, and weakly antagonistic to αβγ and α4β2δ GABAARs.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥437 有现货
100MG 获取报价 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    THIP
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    THIP has a strong affinity for the δ subunit of GABAA receptors. THIP is a functionally selective GABAAR ligand, agonistic to α4β1δ, α4β3δ, and weakly antagonistic to αβγ and α4β2δ GABAARs.
  • 产品描述
    THIP has a strong affinity for the δ subunit of GABAA receptors. THIP is a functionally selective GABAAR ligand, agonistic to α4β1δ, α4β3δ, and weakly antagonistic to αβγ and α4β2δ GABAARs.
  • 同义词
    Gaboxadol; Gaboxadolum
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    PPARγ
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    64603-91-4
  • 分子量
    140.1
  • 分子式
    C6H8N2O2
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    Oc1noc2CNCCc12
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Rasmus K Petersen, et al. Pharmacophore-driven identification of PPARγ agonists from natural sources. J Comput Aided Mol Des. 2011 Feb;25(2):107-16.
产品手册
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