Su1498
CAS No. 168835-82-3
Su1498 ( SU-1498; SU 1498; SU1498; Tyrphostin SU 1498 )
产品货号. M17363 CAS No. 168835-82-3
SU 1498 is a selective inhibitor of the receptor tyrosine kinase VEGF receptor 2 (VEGFR2, aka FLK1; IC50 = 700 nM).
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥381 | 有现货 |
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5MG | ¥583 | 有现货 |
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10MG | ¥988 | 有现货 |
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25MG | ¥1887 | 有现货 |
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50MG | ¥2803 | 有现货 |
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100MG | ¥4155 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Su1498
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述SU 1498 is a selective inhibitor of the receptor tyrosine kinase VEGF receptor 2 (VEGFR2, aka FLK1; IC50 = 700 nM).
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产品描述SU 1498 is a selective inhibitor of the receptor tyrosine kinase VEGF receptor 2 (VEGFR2, aka FLK1; IC50 = 700 nM), having negligible activity at several other serine/threonine and tyrosine kinases.1, 2 It effectively blocks signaling through VEGFR2 both in vitro and in vivo.1, 3 SU 1498 is used to study the role of VEGFR2 signaling in diverse processes, including angiogenesis, tumor growth, neural progenitor cell survival, and neuroregeneration.
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同义词SU-1498; SU 1498; SU1498; Tyrphostin SU 1498
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通路Others
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靶点Other Targets
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受体VEGFR2
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研究领域——
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适应症——
化学信息
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CAS Number168835-82-3
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分子量390.53
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分子式C25H30N2O2
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纯度98%
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溶解度DMSO : ≥ 150 mg/mL. 384.10 mM
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SMILESO=C(/C(=C/c1cc(C(C)C)c(O)c(C(C)C)c1)/C#N)NCCCc1ccccc1
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化学全称(2E)-2-cyano-3-[4-hydroxy-3,5-bis(1-methylethyl)phenyl]-N-(3-phenylpropyl)-2-propenamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1: Gawlak G, et al.Am J Physiol Lung Cell Mol Physiol. 2016 Jun 1;310(11):L1062-70.
产品手册
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