• 咨询热线
    客服服务热线 13671568941/15317326293
  • 在线咨询
  • 微信客服
    微信客服
  • 公众号
    扫码关注公众号

Stiripentol

CAS No. 49763-96-4

Stiripentol ( BCX2600 )

产品货号. M18654 CAS No. 49763-96-4

Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 μM and IC50 of 1.58/3.29 μM, respectively.

纯度: 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥381 有现货
10MG ¥608 有现货
25MG ¥1239 有现货
50MG ¥1758 有现货
100MG ¥2973 有现货
200MG ¥4398 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Stiripentol
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 μM and IC50 of 1.58/3.29 μM, respectively.
  • 产品描述
    Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 μM and IC50 of 1.58/3.29 μM, respectively.
  • 同义词
    BCX2600
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    CYP3A4; CYP2C19
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    49763-96-4
  • 分子量
    234.29
  • 分子式
    C14H18O3
  • 纯度
    98%
  • 溶解度
    DMSO : 150 mg/mL 640.23 mM;
  • SMILES
    CC(C)(C)C(O)\C=C\c1ccc2OCOc2c1
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Giraud C, et al. In vitro and in vivo inhibitory effect of stiripentol on clobazam metabolism.Drug Metab Dispos. 2006 Apr;34(4):608-11. Epub 2006 Jan 13.
产品手册
关联产品
  • BDC2.5 mimotope 1040...

    This is a effectively agonistic peptide (mimotope) for diabetogenic T cell clone BDC2.5. It can stimulate BDC2.5 cells with cells showing good response to this mimotope. 1040-31 peptide is specific for BDC2.5 TCR Tg+ (transgenic) T cells. This peptide is also known as p31.

  • 3,4-Dihydroxyphenyle...

    3, 4-Dihydroxyphenylethanol is an active ingredient extracted from the olive.

  • Methyl nomilinate

    Methyl nomilinate from citrus can modulate cell cycle regulators to induce cytotoxicity in human colon cancer (SW480) cells in vitro.