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SP-13786
CAS No. 1448440-52-5
SP-13786 ( UAMC-1110 )
产品货号. M21138 CAS No. 1448440-52-5
SP-13786 is an inhibitor of fibroblast activation protein (FAP) (IC50 : 3.2 nM); also inhibits prolyl oligopeptidase (PREP) ( IC50 : 1.8 μM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥1037 | 有现货 |
|
| 5MG | ￥1717 | 有现货 |
|
| 10MG | ￥2535 | 有现货 |
|
| 25MG | ￥4277 | 有现货 |
|
| 50MG | ￥6180 | 有现货 |
|
| 100MG | ￥8667 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称SP-13786
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述SP-13786 is an inhibitor of fibroblast activation protein (FAP) (IC50 : 3.2 nM); also inhibits prolyl oligopeptidase (PREP) ( IC50 : 1.8 μM).
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产品描述SP-13786 is an inhibitor of fibroblast activation protein (FAP) (IC50 : 3.2 nM); also inhibits prolyl oligopeptidase (PREP) ( IC50 : 1.8 μM).
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同义词UAMC-1110
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通路Others
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靶点Other Targets
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受体FAP
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研究领域——
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适应症——
化学信息
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CAS Number1448440-52-5
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分子量344.32
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分子式C17H14F2N4O2
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纯度>98% (HPLC)
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溶解度DMSO:100 mg/mL (290.43 mM; Need ultrasonic)
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SMILESN#CC1CC(F)(F)CN1C(=O)CNC(=O)c1ccnc2ccccc12
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Jansen K Heirbaut L Verkerk R et al. Extended Structure–Activity Relationship and Pharmacokinetic Investigation of (4-Quinolinoyl)glycyl-2-cyanopyrrolidine Inhibitors of Fibroblast Activation Protein (FAP)[J]. Journal of Medicinal Chemistry 2014 57(7):3053-3074.
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