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Pridopidine
CAS No. 346688-38-8
Pridopidine ( ACR16;FR-310826;ASP-2314;Huntexil )
产品货号. M14190 CAS No. 346688-38-8
Pridopidine (ACR16, FR-310826, ASP-2314, Huntexil) is a specific dopamine stabilizer without no partial agonism.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥275 | 有现货 |
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| 5MG | ￥551 | 有现货 |
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| 10MG | ￥956 | 有现货 |
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| 25MG | ￥1855 | 有现货 |
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| 50MG | ￥2778 | 有现货 |
|
| 100MG | ￥4026 | 有现货 |
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| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Pridopidine
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Pridopidine (ACR16, FR-310826, ASP-2314, Huntexil) is a specific dopamine stabilizer without no partial agonism.
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产品描述Pridopidine (ACR16, FR-310826, ASP-2314, Huntexil) is a specific dopamine stabilizer without no partial agonism; shows robust dose-dependent striatal D2 occupancy with ED50 of 18.99 mg/kg s.c. in vivo, shows high in vivo D2 receptor occupancy, antipsychotic-like efficacy, and low potential for motor side effects in rats.Parkinson Disease Discontinued
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同义词ACR16;FR-310826;ASP-2314;Huntexil
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通路GPCR/G Protein
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靶点Dopamine Receptor
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受体Dopamine Receptor
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研究领域Neurological Disease
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适应症Parkinson Disease
化学信息
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CAS Number346688-38-8
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分子量281.41
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分子式C15H23NO2S
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纯度>98% (HPLC)
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溶解度DMSO : 50 mg/mL 177.68 mM
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SMILESO=S(C1=C(F)C(C2CCN(CC)CC2)=CC=C1)(C)=O
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化学全称4-(3-(methylsulfonyl)phenyl)-1-propylpiperidin
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Natesan S, et al. J Pharmacol Exp Ther. 2006 Aug;318(2):810-8.
2. Nilsson M, et al. Prog Neuropsychopharmacol Biol Psychiatry. 2004 Jul;28(4):677-85.
3. Seeman P, et al. Synapse. 2009 Oct;63(10):930-4.
4. Pettersson F, et al. J Med Chem. 2010 Mar 25;53(6):2510-20.
2. Nilsson M, et al. Prog Neuropsychopharmacol Biol Psychiatry. 2004 Jul;28(4):677-85.
3. Seeman P, et al. Synapse. 2009 Oct;63(10):930-4.
4. Pettersson F, et al. J Med Chem. 2010 Mar 25;53(6):2510-20.
产品手册
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