PFK-015 ( PFK015; PFK 015; PFK015. )

产品货号. M18553 CAS No. 4382-63-2

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产品名称

PFK-015
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

PFK-015 is an effective inhibitor of PFKFB3 (IC50: 110 nM) and inhibits PFKFB3 activity in Y cells (IC50: 20 nM).
产品描述

PFK-015 is a potent inhibitor of PFKFB3. The preliminary results in a U87GM xenograft model have shown that PFK-015 has comparable activity to Temozolomide. PFK-015 inhibits glucoseuptake by tumors.
同义词

PFK015; PFK 015; PFK015.
通路

Others
靶点

Other Targets
受体

PFKFB3
研究领域

Cancer
适应症

——

1. Clem BF, et al. Mol Y Ther. 2013, 12(8), 1461-1470.

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