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Ocinaplon

CAS No. 96604-21-6

Ocinaplon ( DOV 273547 )

产品货号. M27674 CAS No. 96604-21-6

Ocinaplon is a GABAA receptors modulator.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥721 有现货
10MG ¥1256 有现货
25MG ¥2535 有现货
50MG ¥3791 有现货
100MG ¥5451 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Ocinaplon
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Ocinaplon is a GABAA receptors modulator.
  • 产品描述
    Ocinaplon is a GABAA receptors modulator.(In Vivo):In rats, ocinaplon produces significant muscle relaxation, ataxia, and sedation only at doses >25-fold higher than the minimum effective dose (3.1 mg/kg) in the Vogel "conflict" test.
  • 同义词
    DOV 273547
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    P2X7
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    96604-21-6
  • 分子量
    301.3
  • 分子式
    C17H11N5O
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    O=C(c1cnn2c(ccnc12)-c1ccncc1)c1ccccn1
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Hopper AT, et al. Synthesis and Characterization of the Novel Rodent-Active and CNS-Penetrant P2X7 Receptor Antagonist Lu AF27139. J Med Chem. 2021;64(8):4891-4902.
产品手册
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