Ocinaplon
CAS No. 96604-21-6
Ocinaplon ( DOV 273547 )
产品货号. M27674 CAS No. 96604-21-6
Ocinaplon is a GABAA receptors modulator.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥721 | 有现货 |
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10MG | ¥1256 | 有现货 |
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25MG | ¥2535 | 有现货 |
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50MG | ¥3791 | 有现货 |
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100MG | ¥5451 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Ocinaplon
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Ocinaplon is a GABAA receptors modulator.
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产品描述Ocinaplon is a GABAA receptors modulator.(In Vivo):In rats, ocinaplon produces significant muscle relaxation, ataxia, and sedation only at doses >25-fold higher than the minimum effective dose (3.1 mg/kg) in the Vogel "conflict" test.
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同义词DOV 273547
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通路Others
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靶点Other Targets
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受体P2X7
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研究领域——
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适应症——
化学信息
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CAS Number96604-21-6
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分子量301.3
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分子式C17H11N5O
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C(c1cnn2c(ccnc12)-c1ccncc1)c1ccccn1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Hopper AT, et al. Synthesis and Characterization of the Novel Rodent-Active and CNS-Penetrant P2X7 Receptor Antagonist Lu AF27139. J Med Chem. 2021;64(8):4891-4902.
产品手册
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