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Nortadalafil
CAS No. 171596-36-4
Nortadalafil ( Demethyl Tadalafil )
产品货号. M20552 CAS No. 171596-36-4
Nortadalafil is demethyl Tadalafil which is a PDE5 inhibitor treating erectile dysfunction (ED) ; and under the name Adcirca for the treatment of pulmonary arterial hypertensio.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥356 | 有现货 |
|
| 5MG | ￥583 | 有现货 |
|
| 10MG | ￥915 | 有现货 |
|
| 25MG | ￥1725 | 有现货 |
|
| 50MG | ￥3013 | 有现货 |
|
| 100MG | ￥4836 | 有现货 |
|
| 200MG | ￥6861 | 有现货 |
|
| 500MG | ￥10206 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Nortadalafil
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Nortadalafil is demethyl Tadalafil which is a PDE5 inhibitor treating erectile dysfunction (ED) ; and under the name Adcirca for the treatment of pulmonary arterial hypertensio.
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产品描述Nortadalafil is demethyl Tadalafil which is a PDE5 inhibitor treating erectile dysfunction (ED) ; and under the name Adcirca for the treatment of pulmonary arterial hypertensio.
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同义词Demethyl Tadalafil
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通路Angiogenesis
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靶点PDE
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受体PDE5
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研究领域——
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适应症——
化学信息
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CAS Number171596-36-4
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分子量375.38
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分子式C21H16N3O4
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纯度>98% (HPLC)
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溶解度DMSO:50 mg/mL (133.20 mM)
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SMILESO=C1CNC(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@H](N12)c1ccc2OCOc2c1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Takahiro R Nakamura S Kohno H et al. Contribution of CYP3A Isoforms to Dealkylation of PDE5 Inhibitors: A Comparison between Sildenafil N-Demethylation and Tadalafil Demethylenation[J]. Biological & Pharmaceutical Bulletin 2015 38(1):58-65.
产品手册
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