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Milveterol
CAS No. 652990-07-3
Milveterol ( GSK 159797 )
产品货号. M15483 CAS No. 652990-07-3
Milveterol (GSK 159797) 是一种有效的、选择性长效 β2 肾上腺素受体激动剂，在细胞检测中 pEC50 为 10.2。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 25MG | ￥9858 | 有现货 |
|
| 50MG | ￥12834 | 有现货 |
|
| 100MG | ￥15750 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Milveterol
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Milveterol (GSK 159797) 是一种有效的、选择性长效 β2 肾上腺素受体激动剂，在细胞检测中 pEC50 为 10.2。
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产品描述Milveterol (GSK 159797) is a potent, selective long-acting β2 adrenoceptor agonist with pEC50 of 10.2 in cell-based assays, displays good β2/β1 selectivity (>300-fold); demonstrates high potency in vitro and long duration of action in a guinea pig model of bronchoprotection.Asthma Phase 2 Discontinued.
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体外实验——
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体内实验——
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同义词GSK 159797
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通路GPCR/G Protein
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靶点Adrenergic Receptor
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受体Adrenergic Receptor
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研究领域Inflammation/Immunology
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适应症Asthma
化学信息
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CAS Number652990-07-3
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分子量435.524
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分子式C25H29N3O4
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纯度>98% (HPLC)
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溶解度——
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SMILESC1=CC=C(C=C1)C(CNC2=CC=C(C=C2)CCNCC(C3=CC(=C(C=C3)O)NC=O)O)O
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化学全称N-(2-hydroxy-5-((R)-1-hydroxy-2-((4-(((R)-2-hydroxy-2-phenylethyl)amino)phenethyl)amino)ethyl)phenyl)formamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
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Guanabenz acetate
一种 α2 肾上腺素受体，用作抗高血压化合物。
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Saterinone
Saterinone is a potent and selective phosphodiesterase III inhibitor and a potent antagonist of the vascular α-1-adrenoceptor. Saterinone has vasodilatory properties and can be used in the acute treatment of chronic heart failure. Saterinone inhibited crude cAMP phosphodiesterase (PDE) activity in guinea pig right ventricular homogenates The ic50 value is 2.3 × 10(-5) mol/l.
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Arotinolol hydrochlo...
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