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Metoclopramide
CAS No. 364-62-5
Metoclopramide ( Metoclopramide, Afipran, Maxolon, Reglan, Maxeran, Cerucal )
产品货号. M14253 CAS No. 364-62-5
A potent dopamine D2 receptor antagonist with Ki of 28 nM; also is a mixed 5-HT3 receptor antagonist/5-HT4 receptor agonist.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 100MG | ￥446 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Metoclopramide
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述A potent dopamine D2 receptor antagonist with Ki of 28 nM; also is a mixed 5-HT3 receptor antagonist/5-HT4 receptor agonist.
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产品描述A potent dopamine D2 receptor antagonist with Ki of 28 nM; also is a mixed 5-HT3 receptor antagonist/5-HT4 receptor agonist; commonly used to treat nausea and vomiting caused by chemotherapy.Chemotherapeutic Agents Phase 2 Discontinued
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同义词Metoclopramide, Afipran, Maxolon, Reglan, Maxeran, Cerucal
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通路GPCR/G Protein
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靶点Dopamine Receptor
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受体dopamine D2
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研究领域Cancer
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适应症Chemotherapeutic
化学信息
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CAS Number364-62-5
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分子量299.80
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分子式C14H22ClN3O2
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纯度>98% (HPLC)
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溶解度DMSO: ≥ 41 mg/mL
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SMILESO=C(NCCN(CC)CC)C1=CC(Cl)=C(N)C=C1OC
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化学全称Benzamide, 4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-methoxy-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Matsui A, et al. J Pharmacol Exp Ther. 1998 Nov;287(2):725-32.
2. Tonini M, et al. Pharmacol Res. 1995 May;31(5):257-60.
3. Bateman DN, et al. Br J Clin Pharmacol. 1978 Nov;6(5):401-7.
2. Tonini M, et al. Pharmacol Res. 1995 May;31(5):257-60.
3. Bateman DN, et al. Br J Clin Pharmacol. 1978 Nov;6(5):401-7.
产品手册
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